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4

抑制剂 & 化合物

2

天然产物

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Cat. No. Product Name Target Signaling Pathways
T40060 Nicotinamide riboside malate

Nicotinamide riboside malate is an orally active NAD+ precursor that elevates NAD+ levels and stimulates the activity of SIRT1 and SIRT3. Functioning as a vitamin B3 (niacin) source, it augments oxidative metabolism and provides protection against metabolic abnormalities induced by a high-fat diet. Additionally, Nicotinamide riboside malate mitigates cognitive decline in a genetically modified mouse model of Alzheimer's disease.
T40059 Nicotinamide riboside tartrate

Nicotinamide riboside tartrate (NRT) is an oral NAD+ precursor that raises NAD+ levels, activates SIRT1 and SIRT3, and serves as a vitamin B3 (niacin) source. NRT also improves oxidative metabolism and protects against metabolic abnormalities induced by a high-fat diet. Furthermore, NRT mitigates cognitive decline in a transgenic mouse model of Alzheimer's disease.
T33663 Nicotinamide Riboside Triflate

SRT 647 Triflate,SRT 647,Nicotinamide Riboside,Nicotinamide Ribose,SRT-647,SRT647,SRT647 Triflate,SRT-647 Triflate

Sirtuin Chromatin/Epigenetic; DNA Damage/DNA Repair
Nicotinamide Riboside Triflate (SRT647 Triflate) 是一种天然NAD前体,可增加NAD水平,可增强氧化代谢并防止高脂肪饮食引起的肥胖,KE 激活SIRT3可防止噪音引起的听力损失,可用于研究肌肉萎缩。
T12854 SBI-797812

NAMPT Metabolism
SBI-797812 是在结构上类似于活性位点定向的 NAMPT 抑制剂的化合物,能够阻断这些抑制剂与 NAMPT 的结合。 它将 NAMPT 反应平衡转向 NMN 形成,提高 NAMPT 对 ATP 的亲和力,稳定 His247 处的磷酸化 NAMPT,增加焦磷酸盐副产物的消耗,并通过 NAD+钝化反馈抑制。

化合物

Nicotinamide riboside malate
Cat.No: T40060
Synonym:
Target:
Nicotinamide riboside tartrate
Cat.No: T40059
Synonym:
Target:
Nicotinamide Riboside Triflate
Cat.No: T33663
Synonym: SRT 647 Triflate,SRT 647,Nicotinamide Riboside,Nicotinamide Ribose,SRT-647,SRT647,SRT647 Triflate,SRT-647 Triflate
Target: Sirtuin
SBI-797812
Cat.No: T12854
Synonym:
Target: NAMPT
Cat. No. Product Name Target Signaling Pathways
T13795 Nicotinamide riboside

Sirtuin Chromatin/Epigenetic; DNA Damage/DNA Repair
Nicotinamide riboside 是维生素 B3 的来源,可以增强氧化代谢并防止高脂肪饮食诱导的代谢异常。它是具有口服活性的 NAD+的前体,增加 NAD+水平并激活SIRT1和SIRT3,可用于研究阿尔茨海默氏病的认知退化。
T6220 Nicotinamide riboside chloride

烟酰胺核糖氯酸盐,烟酰胺核苷

Sirtuin; Endogenous Metabolite Chromatin/Epigenetic; DNA Damage/DNA Repair; Metabolism
Nicotinamide riboside Chloride 是维生素 B3 的来源,可以增强氧化代谢并防止高脂肪饮食诱导的代谢异常。它是具有口服活性的 NAD+的前体,增加 NAD+水平并激活SIRT1和SIRT3,可用于研究阿尔茨海默氏病的认知退化。

天然产物

Nicotinamide riboside
Cat.No: T13795
Synonym:
Target: Sirtuin
Nicotinamide riboside chloride
Cat.No: T6220
Synonym: 烟酰胺核糖氯酸盐,烟酰胺核苷
Target: Sirtuin, Endogenous Metabolite
TargetMol Loading
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